selected publications
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academic article
- In Vitro and In Vivo Pharmacological Characterization of a Novel TRPM8 Inhibitor Chemotype Identified by Small-Scale Preclinical Screening. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. 2070-2087. 2022
- New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 114435. 2022
- ß-Lactam TRPM8 antagonist RGM8-51 displays analgesic activity in different animal models. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. 2692-2716. 2022
- Phenylalanine-derived beta-Lactam TRPM8 modulators. Configuration effect on the antagonist activity. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. 2370-2392. 2021
- Exploration of TRPM8 Binding Sites by Carboline-based Antagonists and Their In Vitro Characterization and in Vivo Analgesic Activities. JOURNAL OF MEDICINAL CHEMISTRY. 9672-9694. 2020
- Highly functionalized ß-lactams and 2-ketopiperazines as TRPM8 antagonists with antitumor and antiallodynic activity.. SCIENTIFIC REPORTS. 14154-14165. 2020
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congress communication
- Identificación y Caracterización de nuevos moduladores de TRPM8. 2022
- Amino acid-derived ß¿lactams: TRPM8 antagonists with analgesic activity in different pain models. 2022
- Development of a compound as neurocosmetic ingredient to alleviate allodynia symptoms induced by chemotherapy- 2022
- Discovery of new TRPM8 modulators and their therapeutic potential 2022
- New chiral heterocyclic amino acid derivatives as TRPM8 antagonists. 2022
- New chiral heterocyclic compounds with potent TRPM8 antagonist activity 2022
- Identificación y Caracterización de nuevos moduladores de TRPM8. 2021
- Identification and characterization of new TRPM8 modulators. 2021
- The TRPM8 antagonist RGM8¿51 displays analgesic activity in different pain models. 2021
- ¿Identificación y caracterización de nuevos moduladores del canal TRPM8 2021
- ß¿Lactam TRPM8 antagonists with analgesic activity in different pain models 2021
- Identificación y caracterización de nuevos moduladores del canal TRPM8 2020
- Identificación y caracterización de nuevos moduladores del canal TRPM8 2020
- Identificación y caracterización de nuevos moduladores de TRPM8 2019
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thesis